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S. Clementi, G. Cruciani, M. Pastor and T. Lundstedt, “Series Design in Synthetic Chemistry,” In: F. Gualtieri, Ed., New Trends in Synthetic Medicinal Chemistry, Vol. 7, Wiley-VCH, Weinheim, 2000, pp. 17-37. doi:10.1002/9783527613403.ch2

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