Article citationsMore>>

Chadha, N. and Silakari, O. (2017) Indoles as Therapeutics of Interest in Medicinal Chemistry: Bird’s Eye View. European Journal of Medicinal Chemistry, 134, 159-184.
https://doi.org/10.1016/j.ejmech.2017.04.003

has been cited by the following article:

• TITLE: A Remarkable Regioselective C3-Allylation of Indoles Using Potassium Allyltrifluoroborate under Palladium Catalysis

  AUTHORS: Mohammad Al-Masum, Milton Kumar Kundu, Md Shahin Reza

  KEYWORDS: Indole C3-Allylation, Regioselective Functionalization Potassium Allyltrifluoroborate, Palladium Catalysis, PdCl2(dtbpf) Catalyst

  JOURNAL NAME: International Journal of Organic Chemistry, Vol.16 No.1, March 27, 2026

  ABSTRACT: We report a new and efficient regioselective C3 allylation of indoles using potassium allyltrifluoroborate under PdCl2(dtbpf) catalysis and microwave assisted conditions. The method offers operational simplicity, high regioselectivity, good to excellent yields, and broad substrate compatibility. This study establishes potassium allyltrifluoroborate as a practical allylating reagent for indole functionalization and expands its applicability in synthetic organic chemistry.