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Jalilian, A.R., Sattari, S., Bineshmarvasti, M., Shafiee, A. and Daneshtalab M. (2000) Synthesis and in vitro antifungal and cytotoxicity evaluation of thiazolo-4H-1,2,4-triazoles and 1,2,3-thiadiazolo-4H-1,2,4-triazoles. Arch Pharm (Weinheim), 333, 347-354. doi:10.1002/1521-4184(200010)333:10<347::AID-ARDP347>3.0.CO;2-6

has been cited by the following article:

• TITLE: Synthesis and in vitro antibacterial evaluation of some thiosemicarbazides and thiosemicarbazones

  AUTHORS: Morasa Sheikhy, Amir R. Jalilian, Aytak Novinrooz, Farahnaz Motamedi-Sedeh

  KEYWORDS: Synthesis; Antibacterial; Thiosemicarbazides; Thiosemi-carbazones

  JOURNAL NAME: Journal of Biomedical Science and Engineering, Vol.5 No.2, February 28, 2012

  ABSTRACT: In the present study various thiosemicarbazides and thiosemicarbazones were synthesized and screened for their antimicrobial activity. Among the ligands tested, compounds 1, 3, 4 and 5 demonstrated inhibitory effects at 0.4 - 0.5 μM concentrations against E. coli while 1-(4-fluorobenzoyl)-N4-ethyl-thiosemicar-bazide (3) demonstrated the maximum inhibitory effective compound against E. coli, also possessing high water solubility. Instead, compound 3 demonstrated weak antibiotic effects against S. aurous while compounds 4 - 6 demonstrated significant antibacterial effects at 0.4 - 0.42 μM against the latter organism. Chloramphenicol was used as the positive control.