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Dragovich, P.S., Pillow, T.H., Blake, R.A., Sadowsky, J.D., Adaligil, E., Adhikari, P., Chen, J., Corr, N., Dela Cruz-Chuh, J., Del Rosario, G., Fullerton, A., Hartman, S.J., Jiang, F., Kaufman, S., Kleinheinz, T., Kozak, K.R., Liu, L., Lu, Y., Mulvihill, M.M., Murray, J.M., O’Donohue, A., Rowntree, R.K., Sawyer, W.S., Staben, L.R., Wai, J., Wang, J., Wei, B., Wei, W., Xu, Z., Yao, H., Yu, S.F., Zhang, D., Zhang, H., Zhang, S., Zhao, Y., Zhou, H. and Zhu, X. (2021) Antibody-Mediated Delivery of Chimeric BRD4 Degraders. Part 2: Improvement of in Vitro Antiproliferation Activity and in Vivo Antitumor Efficacy. Journal of Medicinal Chemistry, 64, 2576-2607.
https://doi.org/10.1021/acs.jmedchem.0c01846

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