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Haouz, A., Vanheusden, V., Munier-Lechman, H., Froeyen, M., Herdewijn, P., Van Calenbergh, S. and Delarue, M. (2003) Enzymatic and Structural Analysis of Inhibitors Designed against Mycobacterium tuberculosis Thymidylate Kinase: New Insights into the Phosphoryl Transfer Mechanism. The Journal of Biological Chemistry, 278, 4963-4971.
https://doi.org/10.1074/jbc.M209630200

has been cited by the following article:

• TITLE: Nucleosides 10: Synthesis of New Derivatives of Pyrimidine and Fused Pyrimidine Nucleosides of Expected Biological Activity

  AUTHORS: Laila M. Break, Mosselhi A. M. Mohamed, Ohoud A. A. Al-Thubaiti, Fatma E. M. Eibaih

  KEYWORDS: Synthesis, Nucleosides, Pyrimidines, Fused Pyrimidines Heterocycles, Biological Activity

  JOURNAL NAME: International Journal of Organic Chemistry, Vol.9 No.3, July 11, 2019

  ABSTRACT: Pyrimidines, such as 6-amino-2-thio and 2-methylthiouracils and fused pyrimidines, such as thienopyrimidines reacted with 1-O-acetyl-2,3,5-tri-O- benzoyl-β-D-ribofuranose to get new derivatives of the corresponding nucleosides. The obtained protected nucleosides were deprotected by methanolic sodium methoxide to get the corresponding free uracil and thienopyrimidine nucleosides. The new nucleosides formed were tested for biological activity against some of microorganism (some fungi and bacteria species). Some of the tested products showed moderate activity and the results were reported.