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Wang, X., Shui, Q., Tang, C., Liu, S., Ouyang, Q. and Shi, H. Azilsartan Crystal Form and Its Preparation and Application of the Same. Chinese Patent CN103880829A.

has been cited by the following article:

• TITLE: Crystal Type Iof Azilsartan Polymorphs: Preparation and Analysis

  AUTHORS: Yuhua Ge, Tingting Li, Jingjing Cheng

  KEYWORDS: Azilsartan, Single Crystal Diffraction, Powder Diffraction, Solubility, Stability

  JOURNAL NAME: Journal of Crystallization Process and Technology, Vol.6 No.1, January 28, 2016

  ABSTRACT: Azilsartan (2-ethoxy-1-([2’-(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)biphenyl-4-yl]methyl)-1H-benzimidazole-7-carboxylic acid) is a new angiotensin II receptor antagonist used in the treatment of hypertension. This paper describes the preparation of type I crystal and its single crystal diffraction data, the comparison of the powder diffraction data for both type I and II crystals as well as their stability and solubility in methanol.